Pharmaceutical intermediates

Jingkangen Biomedical provides different types of Pharmaceutical intermediates ranging from milligrams to kilograms scale (1000kg) with high quality and competitive prices.

View More +

Home - Products-JKN Signaling Pathways-Selpercatinib

Selpercatinib

CAS:

2152628-33-4

Cat No:

JKN03215

Purity:

98%

Inquire Now + Next Product +

Note: All products of the company are for scientific research only, and do not provide products and services for any individual

Product Description

CAS	2152628-33-4	Cat No	JKN03215
Name	Selpercatinib
Synonyms	LOXO-292
Smiles	CC(C)(COC1=CN2C(=C(C=N2)C#N)C(=C1)C3=CN=C(C=C3)N4CC5CC(C4)N5CC6=CN=C(C=C6)OC)O
Chemical Name	6-(2-hydroxy-2-methylpropoxy)-4-[6-[6-[(6-methoxypyridin-3-yl)methyl]-3,6-diazabicyclo[3.1.1]heptan-3-yl]pyridin-3-yl]pyrazolo[1,5-a]pyridine-3-carbonitrile
Formula	C29H31N7O3	MWt	525.6
Purity	98%	Storage	Store at 4--8℃
Description	Selpercatinib (LOXO-292; ARRY-192; Retevmo) is a potent,orallybioavailableand highly selective RET (REarrangedduringTransfection) tyrosin kinaseinhibitor with IC50of 14.0 nM, 24.1 nM, and 530.7 nM for RET (WT), RET (V804M), and RET (G810R), respectively.

Product Documents

Products Category

Wuhan Jingkang en Biomedical Technology Co., Ltd.

Tel: +86 137 2013 4139

E-mail: orders@jknbiochem.com

Add.:Room 2120, Office Building 2, No.1 Baisha Fifth Road, Hongshan District, Wuhan City, Hubei Province, China

Get In Touch