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Merestinib

CAS:

1206799-15-6

Cat No:

JKN03224

Purity:

98%

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Product Description

CAS	1206799-15-6	Cat No	JKN03224
Name	Merestinib
Synonyms	LY2801653
Smiles	FC1C([H])=C(C([H])=C([H])C=1OC1C([H])=C2C([H])=NN(C([H])([H])[H])C2=C([H])C=1C1C([H])=NN([H])C=1[H])N([H])C(C1=C([H])C([H])=C(C([H])([H])[H])N(C2C([H])=C([H])C(=C([H])C=2[H])F)C1=O)=O
Chemical Name	N-[3-fluoro-4-[1-methyl-6-(1H-pyrazol-4-yl)indazol-5-yl]oxyphenyl]-1-(4-fluorophenyl)-6-methyl-2-oxopyridine-3-carboxamide
Formula	C30H22F2N6O3	MWt	552.172
Purity	98%	Storage	Store at 4--8℃
Description	Merestinib (LY-2801653) is a novel, potent, orally bioavailable, type-II ATP competitive, slow-off small molecule inhibitor of MET tyrosine kinase with a dissociation constant (Ki) of 2 nM, a pharmacodynamic residence time (Koff) of 0.00132 min(-1) and t1/2 of 525 min.

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Wuhan Jingkang en Biomedical Technology Co., Ltd.

Tel: +86 137 2013 4139

E-mail: orders@jknbiochem.com

Add.:Room 2120, Office Building 2, No.1 Baisha Fifth Road, Hongshan District, Wuhan City, Hubei Province, China

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